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Journal Articles Organic Chemistry Frontiers Year : 2022

Development of novel Gemini-cholesterol analogues for retinoid-related orphan receptors

Uxía Gómez-Bouzó
  • Function : Author
Alioune Fall
  • Function : Author
Judit Osz
  • Function : Author
Yagamare Fall
Hugo Santalla

Abstract

Synthesis of six novel Gemini cholesterol analogues and the binding mode of one of them to RORγ.
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Dates and versions

hal-03745353 , version 1 (04-08-2022)

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Uxía Gómez-Bouzó, Alioune Fall, Judit Osz, Yagamare Fall, Natacha Rochel, et al.. Development of novel Gemini-cholesterol analogues for retinoid-related orphan receptors. Organic Chemistry Frontiers, 2022, 9 (6), pp.1522-1530. ⟨10.1039/D2QO00040G⟩. ⟨hal-03745353⟩
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