Gold(I) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes: towards functionalised azoles
Résumé
Gold(I) catalysed regio-and stereoselective intermolecular hydroamination of internal alkynes was developed for the effective synthesis of a series of (Z)-functionalised vinylazoles under solvent free conditions. The catalytic hydrogenation of the resulting enamines leads to substituted saturated azoles in good yields.
Origine : Fichiers produits par l'(les) auteur(s)
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