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Article Dans Une Revue Tetrahedron Letters Année : 2012

Enantioselective straightforward access to benzo[b]thiophene analogs of azatoxin.

Résumé

Horner-Wadsworth Emmons olefination followed by asymmetric hydrogenation allowed the first synthetic access to the chiral thiotryptophan with good enantiomeric excess. Oxazolidinone formation followed by a Pictet–Spengler condensation provided the benzothiophenic analog of Azatoxin.
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hal-01170195 , version 1 (01-07-2015)

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  • HAL Id : hal-01170195 , version 1

Citer

Stéphanie Gracia, Cédric Marion, Jullien Rey, Florence Popowycz, S Pellet-Rostaing, et al.. Enantioselective straightforward access to benzo[b]thiophene analogs of azatoxin.. Tetrahedron Letters, 2012, 53 (25), pp.3165-3168. ⟨hal-01170195⟩
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