Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid. - Archive ouverte HAL Accéder directement au contenu
Article Dans Une Revue Journal of Organic Chemistry Année : 2008

Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.

Résumé

Reaction of azoles, amides, and sulfonamides in dichloroethane with readily available cyclopropylboronic acid in the presence of copper acetate and sodium carbonate afforded the N-cyclopropyl derivatives in good to excellent yields.

Domaines

Chimie organique

Dates et versions

hal-00770131 , version 1 (04-01-2013)

Identifiants

Citer

Sébastien Bénard, Luc Neuville, Jieping Zhu. Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.. Journal of Organic Chemistry, 2008, 73 (16), pp.6441-4. ⟨10.1021/jo801033y⟩. ⟨hal-00770131⟩
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