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Article Dans Une Revue Bioorganic and Medicinal Chemistry Année : 2011

A specific protein disorder catalyzer of HIV-1 Nef

Résumé

The HIV-1 auxiliary protein Nef is required for the onset and progression of AIDS in HIV-1-infected persons. Here, we have deciphered the mode of action of a second-generation inhibitor of Nef, DLC27-14, presenting a competitive IC50 of

Dates et versions

hal-00662295 , version 1 (23-01-2012)

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Adrien Lugari, Sebastian Breuer, Thibault Coursindel, Sandrine Opi, Audrey Restouin, et al.. A specific protein disorder catalyzer of HIV-1 Nef. Bioorganic and Medicinal Chemistry, 2011, 19, pp.7401-7406. ⟨10.1016/j.bmc.2011.10.051⟩. ⟨hal-00662295⟩
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