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Discovery of novel dengue virus NS5 methyltransferase non-nucleoside inhibitors by fragment-based drug design
Fatiha Benmansour
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Iuni Trist
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Bruno Coutard
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Etienne Decroly
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Gilles Querat
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et al.
Journal articles
hal-02061703v1
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Toscana virus nucleoprotein oligomer organization observed in solution
Amal Baklouti
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Adeline Goulet
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Julie Lichiere
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Bruno Canard
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Remi Charrel
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et al.
Journal articles
hal-01802854v1
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Structural characterization of the N-terminal part of the MERS-CoV nucleocapsid by X-ray diffraction and small-angle X-ray scattering
Nicolas Papageorgiou
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Julie Lichiere
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Amal Baklouti
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Francois Ferron
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Marion Sevajol
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et al.
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hal-01439080v1
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Coxsackievirus B3 protease 3C: expression, purification, crystallization and preliminary structural insights
Stavroula Fili
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Alexandros Valmas
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Magdalini Christopoulou
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Maria Spiliopoulou
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Nikos Nikolopoulos
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Journal articles
hal-01439101v1
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NMR study of non-structural proteins-part I: H-1, C-13, N-15 backbone and side-chain resonance assignment of macro domain from Mayaro virus (MAYV)
Efstathios Melekis
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Aikaterini C. Tsika
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Julie Lichiere
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Christos T. Chasapis
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Irene Margiolaki
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et al.
Journal articles
hal-01438992v1
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mRNA Capping by Venezuelan Equine Encephalitis Virus nsP1: Functional Characterization and Implications for Antiviral Research
Changqing Li
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Jaime Guillen
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Nadia Rabah
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Alexandre Blanjoie
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Francoise Debart
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et al.
Journal articles
hal-01439035v1
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Mutations on VEEV nsP1 relate RNA capping efficiency to ribavirin susceptibility
Nadia Rabah
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Oney Ortega Granda
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Gilles Quérat
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Bruno Canard
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Etienne Decroly
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et al.
Journal articles
hal-03030827v1
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Fluoxetine targets an allosteric site in the enterovirus 2C AAA+ ATPase and stabilizes a ring-shaped hexameric complex
Daniel L Hurdiss
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Priscila El Kazzi
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Lisa Bauer
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Nicolas Papageorgiou
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Francois Ferron
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et al.
Journal articles
hal-03572836v1
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Expression, purification and crystallization of the SARS-CoV macro domain
Hélène Malet
,
Karen Dalle
,
Nicolas Bremond
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Fabienne Tocque
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Stéphanie Blangy
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et al.
Acta Crystallographica Section F: Structural Biology and Crystallization Communications, 2006, 62 (4), pp.405-408. ⟨10.1107/S1744309106009274⟩
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hal-02066254v1
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The Cytotoxic Effect of Apis mellifera Venom with a Synergistic Potential of Its Two Main Components—Melittin and PLA2—On Colon Cancer HCT116 Cell Lines
Carole Yaacoub
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Mariam Rifi
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Dany El-Obeid
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Hiba Mawlawi
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Jean-Marc Sabatier
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et al.
Journal articles
hal-03358045v1
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Rapid incorporation of Favipiravir by the fast and permissive viral RNA polymerase complex results in SARS-CoV-2 lethal mutagenesis
Ashleigh Shannon
,
Barbara Selisko
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Nhung-Thi-Tuyet Le
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Johanna Huchting
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Franck Touret
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et al.
Journal articles
inserm-03052188v1
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Snapshots of ADp-ribose bound to Getah virus macro domain reveal an intriguing choreography
Ana Sofia Ferreira-Ramos
,
Gerlind Sulzenbacher
,
Bruno Canard
,
Bruno Coutard
Journal articles
hal-03160433v1
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High specificity and sensitivity of Zika EDIII-based ELISA diagnosis highlighted by a large human reference panel
Jessica Denis
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Sarah Attoumani
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Patrick Gravier
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Bernard Tenebray
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Annabelle Garnier
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et al.
Journal articles
inserm-02416987v1
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Drugs against SARS‐CoV ‐2: What do we know about their mode of action?
Coralie Valle
,
Baptiste Martin
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Franck Touret
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Ashleigh Shannon
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Bruno Canard
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et al.
Journal articles
hal-03030758v1
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The spike glycoprotein of the new coronavirus 2019-nCoV contains a furin-like cleavage site absent in CoV of the same clade
Bruno Coutard
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Coralie Valle
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Xavier de Lamballerie
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Bruno Canard
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Nabil G Seidah
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et al.
Journal articles
inserm-02517696v1
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The RNA Template Channel of the RNA-Dependent RNA Polymerase as a Target for Development of Antiviral Therapy of Multiple Genera within a Virus Family
Lonneke van Der Linden
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Laia Vives-Adrián
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Barbara Selisko
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Cristina Ferrer-Orta
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Xinran Liu
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et al.
Journal articles
hal-01219259v1
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The methyltransferase domain of the Sudan ebolavirus L protein specifically targets internal adenosines of RNA substrates, in addition to the cap structure
Baptiste Martin
,
Bruno Coutard
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Théo Guez
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Guido Paesen
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Bruno Canard
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et al.
Journal articles
inserm-02416986v1
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Viral Macro Domains Reverse Protein ADP-Ribosylation
Changqing Li
,
Yannick Debing
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Gytis Jankevicius
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Johan Neyts
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Ivan Ahel
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et al.
Journal articles
hal-01439096v1
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Ebola virus L protein harbors a new enzymatic activity involved in the internal methylation of RNAs
Baptiste Martin
,
Coralie Valle
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Bruno Coutard
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Bruno Canard
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Françoise Debart
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et al.
Journal articles
hal-02094423v1
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Antiviral activity of [1,2,3]triazolo[4,5- d ]pyrimidin-7(6 H )-ones against chikungunya virus targeting the viral capping nsP1
Alba Gigante
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Asier Gómez-Sanjuan
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Leen Delang
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Changqing Li
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Oskía Bueno
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et al.
Journal articles
hal-01802837v1
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Single pH buffer refolding screen for protein from inclusion bodies
Bruno Coutard
,
Etienne Danchin
,
Rachid Oubelaid
,
Bruno Canard
,
Christophe Bignon
Journal articles
istex
hal-02649344v1
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Arenavirus Glycan Shield Promotes Neutralizing Antibody Evasion and Protracted Infection
Rami Sommerstein
,
Lukas Flatz
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Melissa M. Remy
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Pauline Malinge
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Giovanni Magistrelli
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et al.
Journal articles
hal-01439028v1
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Optimization of a fragment linking hit toward Dengue and Zika virus NS5 methyltransferases inhibitors
Jessica Hernandez
,
Laurent Hoffer
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Bruno Coutard
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Gilles Quérat
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Philippe Roche
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et al.
Journal articles
inserm-02378768v1
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Conformational plasticity of the VEEV macro domain is important for binding of ADP-ribose
Garyfallia Makrynitsa
,
Dioni Ntonti
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Konstantinos Marousis
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Maria Birkou
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Minos-Timotheos Matsoukas
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et al.
Journal articles
inserm-02416973v1
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Structure and Sequence Requirements for RNA Capping at the Venezuelan Equine Encephalitis Virus RNA 5′ End
Oney Ortega Granda
,
Coralie Valle
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Ashleigh Shannon
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Etienne Decroly
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Bruno Canard
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et al.
Journal articles
hal-03426112v1
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Comparative study of chikungunya Virus-Like Particles and Pseudotyped-Particles used for serological detection of specific immunoglobulin M
Gérald Theillet
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Jérôme Martinez
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Christophe Steinbrugger
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Dimitri Lavillette
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Bruno Coutard
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et al.
Journal articles
inserm-02374934v1
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Fluoxetine Inhibits Enterovirus Replication by Targeting the Viral 2C Protein in a Stereospecific Manner
Lisa Bauer
,
Roberto Manganaro
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Birgit Zonsics
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Jeroen Strating
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Priscila El Kazzi
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et al.
Journal articles
inserm-02416968v1
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First insights into the structural features of Ebola virus methyltransferase activities
Coralie Valle
,
Baptiste Martin
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François Ferron
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Véronique Roig-Zamboni
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Aline Desmyter
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et al.
Journal articles
hal-03334409v1
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Assessment of Dengue virus helicase and methyltransferase as targets for fragment-based drug discovery
Bruno Coutard
,
Etienne Decroly
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Changqing Li
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Andrew Sharff
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Julien Lescar
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et al.
Journal articles
hal-02061701v1
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Development and Evaluation of a duo SARS-CoV-2 RT-qPCR Assay Combining Two Assays Approved by the World Health Organization Targeting the Envelope and the RNA-Dependant RNA Polymerase (RdRp) Coding Regions
Laura Pezzi
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Remi Charrel
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Laetitia Ninove
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Antoine Nougairede
,
Gregory Molle
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et al.
Journal articles
hal-02897091v1
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