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First synthesis of diethyl N-acetyl-glycosamine-1- difluoromethylphosphonate from 2-nitroglycals as phosphate analog

Thierry Delaunay , Thomas Poisson , Philippe Jubault , Xavier Pannecoucke
Journal of Fluorine Chemistry, 2015, 171, pp.56-59. ⟨10.1016/j.jfluchem.2014.10.001⟩
Journal articles hal-01149514v1

Convenient preparation of α-bromo-α-fluoro-β-hydroxy esters building blocks from aldehydes, ketones and lactones

Ludivine Zoute , Gérald Lemonnier , Tanh-Mai Nguyen , Jean-Charles Quirion , Philippe Jubault et al.
Tetrahedron Letters, 2011, 52 (19), pp.2473-2475. ⟨10.1016/j.tetlet.2011.03.014⟩
Journal articles hal-01017744v1

Copper Catalyzed Asymmetric Formation of Enantioenriched Trifluoromethylated Synthons

Poutrel Pauline , Xavier Pannecoucke , Philippe Jubault , Thomas Poisson
Journée scientifique de la Fédération de l'Institut normand de chimie moléculaire, médicinale et macromoléculaire (INC3M), Jun 2019, Caen, France
Conference papers hal-02413289v1

Transition Metal Catalyzed Trifluoromethylthiolation Reaction and Heterocycles Synthesis by C-H Bond Functionalization

Mu-Yi Chen , Xavier Pannecoucke , Philippe Jubault , Tatiana Besset
Journées Nord-Ouest Européennes des Jeunes Chercheurs (JNOEJC 2019), Jun 2019, Rouen, France
Conference papers hal-02413613v1

Recent advances in photocatalyzed reactions using well-defined copper(I) complexes

Mingbing Zhong , Xavier Pannecoucke , Philippe Jubault , Thomas Poisson
Beilstein Journal of Organic Chemistry, 2020, 16, pp.451-481. ⟨10.3762/bjoc.16.42⟩
Journal articles hal-02526176v1
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Pd-Catalyzed Selective Chlorination of Acrylamides at Room Temperature

Mu-Yi Chen , Xavier Pannecoucke , Philippe Jubault , Tatiana Besset
Organic Letters, 2020, 22 (19), pp.7556-7561. ⟨10.1021/acs.orglett.0c02750⟩
Journal articles hal-03025282v1

A Straightforward and Highly Diastereoselective Access to Functionalized Monofluorinated Cyclopropanes via a Michael Initiated Ring Closure Reaction

Thibault Ferrary , Emilie David , Gaëlle Milanole , Tatiana Besset , Philippe Jubault et al.
Organic Letters, 2013, 15 (21), pp.5598-5601. ⟨10.1021/ol402837u⟩
Journal articles hal-02541577v1

[18F]CuCF3 :A[18F]Trifluoromethylating Agent for Arylboronic Acids and Aryl Iodides

Pavel Ivashkin , Gérald Lemonnier , Jonathan Cousin , Vincent Grégoire , Daniel Labar et al.
Chemistry - A European Journal, 2014, 20 (31), pp.9514-9518. ⟨10.1002/chem.201403630⟩
Journal articles istex hal-01149583v1
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N‐Thiocyanato‐2,10‐camphorsultam Derivatives: Design and Applications of Original Electrophilic Thiocyanating Reagents

Mélissa Gao , Martin Vuagnat , Philippe Jubault , Tatiana Besset
European Journal of Organic Chemistry, 2021, 2022 (1), pp.e202101255. ⟨10.1002/ejoc.202101255⟩
Journal articles hal-03744635v1

Stereoselective Synthesis of Terminal Monofluoroalkenes from Trifluoromethylated Alkenes

Pauline Poutrel , Xavier Pannecoucke , Philippe Jubault , Thomas Poisson
Organic Letters, 2020, 22 (12), pp.4858-4863. ⟨10.1021/acs.orglett.0c01701⟩
Journal articles hal-02877369v1
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Pd‐Catalyzed Directed Thiocyanation Reaction by C−H Bond Activation

Mélissa Gao , Mu-Yi Chen , Xavier Pannecoucke , Philippe Jubault , Tatiana Besset et al.
Chemistry - A European Journal, 2020, 22 (19), pp.7556-7561. ⟨10.1002/chem.202003521⟩
Journal articles hal-03004678v1

Recent Progress Toward the Synthesis of Trifluoromethyl- and Difluoromethyl-Substituted Cyclopropanes

Maxence Bos , Thomas Poisson , Xavier Pannecoucke , André B. Charette , Philippe Jubault et al.
Chemistry - A European Journal, 2017, 23 (21), pp.4950-4961. ⟨10.1002/chem.201604564⟩
Journal articles hal-02046262v1

One-step synthesis of highly functionalized monofluorinated cyclopropanes from electron-deficient alkenes.

Pavel Ivashkin , Samuel Couve-Bonnaire , Philippe Jubault , Xavier Pannecoucke
Organic Letters, 2012, 14 (9), pp.2270-2273. ⟨10.1021/ol300687s⟩
Journal articles hal-00996598v1

3,3-gem-Difluorinated-β-lactams: synthesis pathways and applications

Thomas Orbegozo , Fabrice Burel , Philippe Jubault , Xavier Pannecoucke
Tetrahedron, 2013, 69 (20), pp.4015-4039. ⟨10.1016/j.tet.2013.02.043⟩
Journal articles hal-01015779v1
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First efficient synthesis of SF 5 -substituted pyrrolidines using 1,3-dipolar cycloaddition of azomethine ylides with pentafluorosulfanyl-substituted acrylic esters and amides

Ewelina Falkowska , Vincent Tognetti , Laurent Joubert , Philippe Jubault , J.-P. Bouillon et al.
RSC Advances, 2015, 5 (9), pp.6864-6868. ⟨10.1039/c4ra14075c⟩
Journal articles hal-01149543v1

Ethyl dibromofluoroacetate: a versatile reagent for the synthesis of fluorinated molecules

Emilie David , Samuel Couve-Bonnaire , Philippe Jubault , Xavier Pannecoucke
Tetrahedron, 2013, 69 (52), pp.11039-11055. ⟨10.1016/j.tet.2013.10.048⟩
Journal articles hal-01015276v1

Synthesis of functionalized fluorocyclopropanes, difluoromethyl and trifluoromethyl cyclopropanes and applications

Philippe Jubault
Séminaire international, Université du Québec, Oct 2019, Montréal, Canada
Conference papers hal-02412980v1

Copper Catalyzed Asymmetric Formation of Enantioenriched Trifluoromethylated Synthons

Poutrel Pauline , Xavier Pannecoucke , Philippe Jubault , Thomas Poisson
Journées Nord-Ouest Européennes des Jeunes Chercheurs (JNOEJC, 2019), Jun 2019, Rouen, France
Conference papers hal-02413168v1

Catalytic Asymmetric Synthesis of α,α-Difluoromethylated and α-Fluoromethylated Tertiary Alcohols

Wei-Sheng Huang , Marie-Léonie Delcourt , Xavier Pannecoucke , André Charette , Thomas Poisson et al.
Organic Letters, 2019, 21 (18), pp.7509-7513. ⟨10.1021/acs.orglett.9b02792⟩
Journal articles hal-02282518v1

Pd‐Catalyzed Directed Thiocyanation Reaction by C–H Bond Activation

Mélissa Gao , Mu-Yi Chen , Xavier Pannecoucke , Philippe Jubault , Tatiana Besset et al.
Chemistry - A European Journal, 2020, ⟨10.1002/chem.202003521⟩
Journal articles hal-02921268v1

Synthesis and evaluation of a broad range of new chiral phosphine-carbene ligands for asymmetric hydrogenation

Johan Passays , Philippe Jubault , Tahar Ayad , Virginie Ratovelomanana-Vidal , Annie-Claude Gaumont et al.
Tetrahedron: Asymmetry, 2011, 22, pp.562-574. ⟨10.1016/j.tetasy.2011.02.017⟩
Journal articles hal-00606050v1

Catalytic Enantioselective Synthesis of Halocyclopropanes

Amandine Pons , Pavel Ivashkin , Thomas Poisson , André B. Charette , Xavier Pannecoucke et al.
Chemistry - A European Journal, 2016, 22 (18), pp.6239-6242. ⟨10.1002/chem.201600649⟩
Journal articles istex hal-01321309v1

New entries toward the synthesis of OCF3-containing molecules

Tatiana Besset , Philippe Jubault , Xavier Pannecoucke , Thomas Poisson
Organic Chemistry Frontiers, 2016, 3 (8), pp.1004-1010. ⟨10.1039/c6qo00164e⟩
Journal articles hal-01404889v1

Toward the Synthesis of Fluorinated Analogues of HCV NS3/4A Serine Protease Inhibitors Using Methyl α-Amino-β-fluoro-β-vinylcyclopropanecarboxylate as Key Intermediate

Gaëlle Milanole , Floris Andriessen , Gérald Lemonnier , Muriel Sebban , Gaël Coadou et al.
Organic Letters, 2015, 17 (12), pp.2968-2971. ⟨10.1021/acs.orglett.5b01216⟩
Journal articles hal-01179463v1

Synthesis of new pentafluorinated heterocycles

Ewelina Falkowska , J.-P. Bouillon , Philippe Jubault , Xavier Pannecoucke
International Symposium on Fluorine Chemistry (ISFC, 21, 2015) - International Symposium on Fluorous Technologies (ISoFT, 6, 2015), Aug 2015, Côme, Italy
Conference papers hal-02378890v1

Synthesis of fluorinated cyclopropyl amino acid analogues: toward the synthesis of original fluorinated peptidomimetics.

Gaëlle Milanole , Samuel Couve-Bonnaire , Jean-François Bonfanti , Philippe Jubault , Xavier Pannecoucke et al.
Journal of Organic Chemistry, 2013, 78 (2), pp.212-223. ⟨10.1021/jo302222n⟩
Journal articles hal-00996635v1
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Recent Advances for the Direct Introduction of the CF2Me Moiety

Elodie Carbonnel , Thomas Poisson , Philippe Jubault , Xavier Pannecoucke , Tatiana Besset et al.
Frontiers in Chemistry, 2019, 7, pp.111. ⟨10.3389/fchem.2019.00111⟩
Journal articles hal-02121212v1
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Z -Selective Pd-catalyzed 2,2,2-trifluoroethylation of acrylamides at room temperature

Louise Ruyet , Maria Lapuh , Vijay Koshti , Tamás Földesi , Philippe Jubault et al.
Chemical Communications, 2021, 57 (51), pp.6241-6244. ⟨10.1039/D1CC02007B⟩
Journal articles hal-03442521v1

Practical Synthesis of Ethyl 3-Fluoro-1-pyrrole-2-carboxylate: A Key Fragment of a Potent Drug Candidate against Hepatitis B Virus

Adeline René , Maxime Quilan , Yicheng Deng , Yang Cheng , Christopher Teleha et al.
Organic Process Research and Development, 2019, 24 (5), pp.792-801. ⟨10.1021/acs.oprd.9b00382⟩
Journal articles hal-02364011v1

Synthesis of functionalized fluorocyclopropanes, difluoromethyl and trifluoromethyl cyclopropanes and applications

Philippe Jubault
Séminaire international, Université de Sherbrooke, Oct 2019, Sherbrooke, Canada
Conference papers hal-02413237v1