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Straightforward synthesis of indolizidine alkaloid 167B

Stéphanie Gracia , Rudolf Jerpan , S Pellet-Rostaing , Florence Popowycz , Marc Lemaire et al.
Tetrahedron Letters, 2010, 51 (48), pp.6290-6293
Journal articles hal-01167326v1

Efficient C-3 reductive alkylation of 4-hydroxycoumarin by dehydrogenative oxidation of benzylic alcohols through ruthenium catalysis

A. Montagut-Romans , M. Boulven , M. Lemaire , Florence Popowycz
New Journal of Chemistry, 2014, 38 (4), pp.1794-1801. ⟨10.1039/c3nj01517c⟩
Journal articles hal-02639455v1

Hydroxymethylfurfural (HMF) and Glucosyloxymethylfurfural (GMF) in Multi-Component Reactions,

W. Fan , C. Verrier , L. Wang , M. Ahmar , N. Tan J. et al.
Recent Trends in Carbohydrate Chemistry, Synthesis, Structure and Function of Carbohydrates, pp.73-100, 2020, 9780128174678. ⟨10.1016/B978-0-12-817467-8.00002-5⟩
Book sections hal-02110911v1

Regioselective Late-Stage C-3 Functionalization of Pyrazolo[3,4-b]pyridines

Hubert Lavrard , Florence Popowycz
Synthesis: Journal of Synthetic Organic Chemistry, 2018, 50 (05), pp.998-1006. ⟨10.1055/s-0036-1589161⟩
Journal articles hal-02110576v1

Pyrazolo[1,5-a]-1,3,5-triazine as a purine bioisostere: access to potent cyclin-dependent kinase inhibitor (R)-roscovitine analogue.

Florence Popowycz , Guy Fournet , Cédric Schneider , Karima Bettayeb , Yoan Ferandin et al.
Journal of Medicinal Chemistry, 2009, 52 (3), pp.655-63. ⟨10.1021/jm801340z⟩
Journal articles hal-00416036v1

Identification of VKORC1 genotype leading to resistance to tecarfarin.

Matagrin Benjamin , Montagut-Romans Adrien , Damin Marlene , Marc Lemaire , Popowycz Florence et al.
Journal of Clinical Pharmacology, 2014, 54, pp.896-900
Journal articles hal-01149817v1
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One-Pot, Solvent-Free Access to Unsymmetrical Ureas by Palladium-Catalysed Reductive Alkylation Using Molecular Hydrogen

Tharwat Mohy El Dine , Simon Chapron , Marie-Christine Duclos , Nicolas Duguet , Florence Popowycz et al.
European Journal of Organic Chemistry, 2013, 2013 (24), pp.5445-5454. ⟨10.1002/ejoc.201300642⟩
Journal articles hal-03249259v1

Synthesis and antiproliferative evaluation of pyrazolo[1,5-a]-1,3,5-triazine myoseverin derivatives.

Florence Popowycz , Cédric Schneider , Salvatore Debonis , Dimitrios Skoufias , Frank Kozielski et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (9), pp.3471-8. ⟨10.1016/j.bmc.2009.03.007⟩
Journal articles hal-00691448v1

Synthesis and evaluation of thiophenyl derivatives as inhibitors of alkaline phosphatase

L. Chang , D. Le Duy , S. Mébarek , F. Popowycz , S Pellet-Rostaing et al.
Bioorganic and Medicinal Chemistry Letters, 2011, 21 (8), pp.2297-2301. ⟨10.1016/j.bmcl.2011.02.089⟩
Journal articles hal-00692020v1
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Novel Non‐toxic and Non‐hazardous Solvent Systems for the Chemistry of Indoles: Use of a Sulfone‐containing Brønsted Acid Ionic Liquid Catalyst in Butyl Acetate

Ahmed El‐harairy , Y. Qi , Meie Yue , Weigang Fan , Florence Popowycz et al.
ChemCatChem, 2019, 11 (17), pp.4403-4410. ⟨10.1002/cctc.201900784⟩
Journal articles hal-02193181v1

Bromination of 3-substituted benzo[b]thiophenes : access to raloxifen intermediate.

François Liger , S Pellet-Rostaing , Florence Popowycz , Marc Lemaire
Tetrahedron Letters, 2011, 52 (29), pp.3736-3739
Journal articles hal-01168536v1

Reduction of aromatic and aliphatic nitro groups to anilines and amines with hypophosphites associated with Pd/C

Marc Baron , Estelle Métay , Marc Lemaire , Florence Popowycz
Green Chemistry, 2013, 15, pp.1006-1015
Journal articles hal-01179144v1

Enantioselective straightforward access to benzo[b]thiophene analogs of azatoxin.

Stéphanie Gracia , Cédric Marion , Jullien Rey , Florence Popowycz , S Pellet-Rostaing et al.
Tetrahedron Letters, 2012, 53 (25), pp.3165-3168
Journal articles hal-01170195v1

Straightfoward synthesis of 2-acetyl-substituted benzo[b]thiophenes

Julien Debray , Marc Lemaire , Florence Popowycz
SYNLETT, 2013, 24, pp.37-40
Journal articles hal-01146314v1

Non classical route to 2,3-diiodoindole derivatives from indole-2-carboxylic acids,

) A. Putey , F. Popowycz , B. Joseph.
SYNLETT, 2007, pp.419
Journal articles hal-00158992v1

Identification of VKORC1 genotype leading to resistance to tecarfarin

Benjamin Matagrin , Adrien Montagut-Romans , Marlene Damin , Marc Lemaire , Florence Popowycz et al.
Journal of Clinical Pharmacology, 2014, 54 (8), pp.896-900. ⟨10.1002/jcph.332⟩
Journal articles istex hal-02636776v1

Is ultrasound improving the reduction of nitro compounds catalyzed by Pd/C using a mixture of sodium hypophosphite and hypophosphorous acid as reducing agent? An investigation

M. Draye , S. Letort , M. Lejeune , N. Kardos , E. Métay et al.
4th International Symposium on Green Chemistry, May 2017, La Rochelle, France
Conference papers hal-02048846v1

Straightforward Synthesis of Chiral Terpenoid Building Blocks by Ru-Catalyzed Enantioselective Hydrogenation

Johal Ruiz , Philippe Oger , Laurent Soulère , Florence Popowycz
Journal of Organic Chemistry, 2021, ⟨10.1021/acs.joc.1c00677⟩
Journal articles hal-03275385v1
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Synthesis of phospholipids under plausible prebiotic conditions and analogies with phospholipid biochemistry or origin of life studies

Michele Fiore , Carolina Chieffo , Augustin Lopez , Dimitri Fayolle , Johal Ruiz et al.
Astrobiology, In press, ⟨10.1089/ast.2021.0059⟩
Journal articles hal-03591985v1
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Comparative inhibitory effect of prenylated coumarins, ferulenol and ferprenin, contained in the 'poisonous chemotype' of Ferula communis on mammal liver microsomal VKORC1 activity.

Marie-Sophie Louvet , Gilbert Gault , Sébastien Lefebvre , Florence Popowycz , Manon Boulven et al.
Phytochemistry, 2015, 118 (118), pp.124-130. ⟨10.1016/j.phytochem.2015.08.012⟩
Journal articles hal-01577246v1
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Development of an ecofriendly anticoagulant rodenticide based on the stereochemistry of difenacoum

Marlène Damin-Pernik , Bernadette Espana , Stéphane Besse , Isabelle Fourel , Hervé Caruel et al.
Drug Metabolism and Disposition, 2016, 44 (12), pp.1872-1880. ⟨10.1124/dmd.116.071688⟩
Journal articles hal-01608089v1

Reductive alkylation of active methylene compounds with carbonyl derivatives, calcium hydride and a heterogeneous catalyst.

Carole Guyon , Marie-Christine Duclos , Marc Sutter , Estelle Metay , Florence Popowycz et al.
Organic & Biomolecular Chemistry, 2015, 13 (25), pp.7067-7075
Journal articles hal-01313010v1

Diastereoselective Iridium-Catalyzed Amination of Biosourced Isohexides Through Borrowing Hydrogen Methodology

Maiwenn Jacolot , Sylvie Moebs-Sanchez , Florence Popowycz
Journal of Organic Chemistry, 2018, 83 (16), pp.9456-9463. ⟨10.1021/acs.joc.8b01162⟩
Journal articles hal-02110500v1

Functionnalization of α-carbolines at the C-6 position

Cédric Schneider , Gueyrard David , Popowycz Florence , Joseph Benoît , Peter G. Goekjian et al.
Symposium de chimie organique Centre-Auvergne-Limousin Poitou-Charente-SYCOCAL PC (52, 2007), May 2007, La Rochelle, France
Conference papers hal-02381215v1

Direct Amination of Isohexides via Borrowing Hydrogen Methodology: Regio- and Stereoselective Issues

Florian Bahé , Lucie Grand , Elise Cartier , Maiwenn Jacolot , Sylvie Moebs-Sanchez et al.
European Journal of Organic Chemistry, 2020, 2020 (5), pp.599-608. ⟨10.1002/ejoc.201901661⟩
Journal articles hal-02572417v1

Catalytic access to anhydrohexitols and their isomerization

Mathieu Sauthier , Isabelle Suisse , Florence Popowycz , Sylvie Moebs-Sanchez , Maïwenn Jacolot et al.
Carbohydrate Chemistry, 45, Royal Society of Chemistry, pp.305-335, 2021, Carbohydrate Chemistry, ⟨10.1039/9781839164538-00305⟩
Book sections hal-03543793v1
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Advances on Multicomponent Reactions Based on Biomass-Derived Platform Molecules

Jing Xu , Weigang Fan , Florence Popowycz , Yves Queneau , Yanlong Gu et al.
Chinese Journal of Organic Chemistry, 2019, 39 (8), pp.2131-2138. ⟨10.6023/cjoc201904065⟩
Journal articles hal-02279725v1

Synthesis and reactivity of 4-, 5- et 6-azaindoles,

F. Popowycz , J.-Y. Merour , B. Joseph.
Tetrahedron, 2007, pp.63,8689
Journal articles hal-00159016v1

Access to the Paullone system via intramolecular Heck reaction, Helv.

L. Joucla , F. Popowycz , O. Lozach , L. Meijer , B. Joseph. et al.
Chim. Acta, 2007, pp.90, 753
Journal articles hal-00158997v1

Chemoselective functionalization of α-carbolines at 2-, 3-, 4- and 6-positions by Suzuki-Miyaura reaction

Cédric Schneider , Florence Popowycz , Joseph Benoît , Peter G. Goekjian , Gueyrard David et al.
Canadian Chemistry Conference and Exhibition (CSC, 92, 2009), May 2009, Hamilton, Canada
Conference papers hal-02381196v1