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Synthesis, biological evaluation, and in vivo imaging of the first camptothecin-fluorescein conjugate.

Arnaud Chevalier , Martine Dubois , Vadim Le Joncour , Sébastien Dautrey , Céline Lecointre , et al.
Bioconjugate Chemistry, 2013, 24 (7), pp.1119-1133. ⟨10.1021/bc3005304⟩
Journal articles hal-00996547v1

Développement d'outils de ligation chimiosélective

Cyrille Sabot
Séminaire national, Faculté de pharmacie de l'Université de Strasbourg, Sep 2017, Strasbourg, France
Conference papers hal-02391479v1

Synthèse expéditive d'alcaloïdes par double stratégie de synthèse d'hétérocycle par micro-ondes

Cyrille Sabot
Symposium francophone de synthèse totale (SFST, 5, 2015), Jun 2015, Strasbourg, France
Conference papers hal-02389669v1

Investigation of tetrazine reactivity towards C-nucleophiles: pyrazolone-based modification of biomolecules

Kévin Renault , Clément Guillou , Pierre-Yves Renard , Cyrille Sabot
Organic & Biomolecular Chemistry, 2019, 17 (2), pp.388-396. ⟨10.1039/C8OB02108B⟩
Journal articles hal-02329641v1

Kondrat'eva reaction: an irreversible Diels-Alder-based chemoselective ligation ?

Cyrille Sabot
The Missing link biologically driven ligation of carbohydrates and proteins, Jun 2016, Kiel, Germany
Conference papers hal-02380448v1

Metal-free oxidative ring contraction of benzodiazepinones: an entry to quinoxalinones

Hasan Mtiraoui , Kévin Renault , Morgane Sanselme , Moncef Msaddek , Pierre-Yves Renard , et al.
Organic & Biomolecular Chemistry, 2017, 15 (14), pp.3060-3068. ⟨10.1039/C7OB00205J⟩
Journal articles hal-02329806v1

Utilisation du motif 5-alkoxyoxazole en synthèse organique et biorganique

Cyrille Sabot
Journées des Chargés de recherche 1 (CR1) du CNRS, Jun 2015, Paris, France
Conference papers hal-02403947v1

Metal-Free Decarboxylative Hetero-Diels-Alder Synthesis of 3-Hydroxypyridines: A Rapid Access to N-Fused Bicyclic Hydroxypiperidine Scaffolds.

Laurie-Anne Jouanno , Vincent Di Mascio , Vincent Tognetti , Laurent Joubert , Cyrille Sabot , et al.
Journal of Organic Chemistry, 2014, 79 (3), pp.1303-1319. ⟨10.1021/jo402729a⟩
Journal articles hal-00996570v1

Total Synthesis and Structural Revision of Chaetoviridins A

Mehdi Makrerougras , Romain Coffinier , Samuel Oger , Arnaud Chevalier , Cyrille Sabot , et al.
Organic Letters, 2017, 19 (15), pp.4146-4149. ⟨10.1021/acs.orglett.7b02053⟩
Journal articles hal-02046297v1

Covalent Modification of Biomolecules through Maleimide-Based Labeling Strategies

Kévin Renault , J.W. Fredy , Pierre-Yves Renard , Cyrille Sabot
Bioconjugate Chemistry, 2018, 29 (8), pp.2497-2513. ⟨10.1021/acs.bioconjchem.8b00252⟩
Journal articles hal-02024527v1

Total synthesis of chaetoviridin A

Mehdi Makrerougras , Cyrille Sabot , Franck Xavier
Anglo-Norman colloquium on organic chemistry (ANORCQ, 13, 2016), Apr 2016, Rouen, France
Poster communications hal-02370675v1

Photophysical properties of quinoxalin-2(1H)-ones: Application in the preparation of an azide-based fluorogenic probe for the detection of hydrogen sulfide

Kévin Renault , Pierre-Yves Renard , Cyrille Sabot
New Journal of Chemistry, 2017, 41 (18), pp.10432-10437. ⟨10.1039/c7nj01893b⟩
Journal articles hal-02046306v1

5-Alkoxyoxazole –A Versatile Building Block in (Bio)organic Synthesis

Laurie-Anne Jouanno , Kévin Renault , Cyrille Sabot , Pierre-Yves Renard
European Journal of Organic Chemistry, 2016, 2016 (20), pp.3264-3281. ⟨10.1002/ejoc.201600127⟩
Journal articles istex hal-02046218v1

A convenient aminolysis of esters catalyzed by 1,5,7-triazabicyclo[4.4.0]dec-5-ene (TBD) under solvent-free conditions.

C. Sabot , K. Ananda Kumar , S. Meunier , C. Mioskowski
Tetrahedron Letters, 2007, 48, pp.3863-3866
Journal articles hal-00165294v1

Insights on two in situ click chemistry reactions for the synthesis of AChE inhibitors

E. Oueis , Ronco C. , F. Nachon , Cyrille Sabot , Ludovic Jean , et al.
International Meeting on Cholinesterases - Sixth International Conference on Paraoxonases (12, 2015), Sep 2015, Elche, Spain
Conference papers hal-02379142v1

Reaction site-driven regioselective synthesis of AChE inhibitors

Emilia Oueis , Gianluca Santoni , Cyril Ronco , Olga A. Syzgantseva , Vincent Tognetti , et al.
Organic & Biomolecular Chemistry, 2014, 12 (1), pp.156-161. ⟨10.1039/C3OB42109K⟩
Journal articles hal-02335933v1

Diverted Natural Lossen-type Rearrangement for Bioconjugation through in Situ Myrosinase-Triggered Isothiocyanate Synthesis

Jean Wilfried Fredy , Giuliano Cutolo , Benjamin Poret , Reine Nehmé , Marie Hubert-Roux , et al.
Bioconjugate Chemistry, 2019, 30 (5), pp.1385-1394. ⟨10.1021/acs.bioconjchem.9b00153⟩
Journal articles hal-02280045v1

Synthèse totale des chaétoviridines A et révisions structurales

Mehdi Makrerougras , Cyrille Sabot , Xavier Franck
Symposium francophone de synthèse totale (SFST, 7, 2017), Jun 2017, Orsay, France
Poster communications hal-02370810v1

Fluorogenic Behaviour of the Hetero-Diels–Alder Ligation of 5-Alkoxyoxazoles with Maleimides and their Applications

Kévin Renault , Laurie-Anne Jouanno , Antoine Lizzul-Jurse , Pierre-Yves Renard , Cyrille Sabot
Chemistry - A European Journal, 2016, 22 (51), pp.18522-18531. ⟨10.1002/chem.201603617⟩
Journal articles istex hal-02046236v1

Méthode de criblage : identification de catalyseurs de la réaction de Diels-Alder

Cyrille Sabot , Laura Nogueira de Faria Cardoso , Pierre-Yves Renard , Wadih Ghattas , Jean-Pierre Mahy
Journée scientifique du LabEx Chimie des Architectures Moléculaires Multifonctionnelles et des Matériaux (CHARMMMAT, 6, 2018)), Jun 2018, Cachan, France
Conference papers hal-03098307v1

Total synthesis of (±)-17-norcamptothecin, a novel E-ring modified camptothecin

Marie Devert , Cyrille Sabot , Pascale Giboreau , Jean-François Constant , Andrew E. Greene , et al.
Tetrahedron, 2010, 66 (35), pp.7227-7231. ⟨10.1016/j.tet.2010.06.003⟩
Journal articles hal-01658636v1

First enzymatic hydrolysis/thio-Michael addition cascade route to synthesis of AChE inhibitors.

Emilia Oueis , Florian Nachon , Cyrille Sabot , Pierre-Yves Renard
Chemical Communications, 2014, 50 (16), pp.2043-2045. ⟨10.1039/c3cc48871c⟩
Journal articles hal-00996567v1

Synthesis of polysubstituted 3-hydroxypyridines via the revisited hetero-Diels-Alder reaction of 5-alkoxyoxazoles with dienophiles.

Cyrille Sabot , Emilia Oueis , Xavier Brune , Pierre-Yves Renard
Chemical Communications, 2012, 48 (5), pp.768-770. ⟨10.1039/c1cc16562c⟩
Journal articles hal-00996467v1

Thermally controlled decarboxylative [4 + 2] cycloaddition between alkoxyoxazoles and acrylic acid: expedient access to 3-hydroxypyridines.

Laurie-Anne Jouanno , Vincent Tognetti , Laurent Joubert , Cyrille Sabot , Pierre-Yves Renard
Organic Letters, 2013, 15 (10), pp.2530-2533. ⟨10.1021/ol4010195⟩
Journal articles hal-00996416v1

Glycosyltransferase inhibitor engineering and its uses to study plant cell growth

Mathieu Carlier , Thomas Poisson , Cyrille Sabot , Jean-Claude Mollet , Patrice Lerouge , et al.
28èmes Journées du Groupe Français des Glycosciences, May 2022, Branville, France
Poster communications hal-03714242v1
Image document

Maleimide-based metal-free ligation with dienes: a comparative study

Alexis Lossouarn , Kévin Renault , Laëtitia Bailly , Axel Frisby , Patricia Le Nahenec-Martel , et al.
Organic & Biomolecular Chemistry, 2020, 18 (20), pp.3874-3887. ⟨10.1039/D0OB00403K⟩
Journal articles hal-03010566v1

Detection of Biothiols with a Fast-Responsive and Water-Soluble Pyrazolone-Based Fluorogenic Probe

Kévin Renault , Pierre-Yves Renard , Cyrille Sabot
European Journal of Organic Chemistry, 2018, 2018 (46), pp.6494-6498. ⟨10.1002/ejoc.201801157⟩
Journal articles hal-02024529v1

From Synthetic Methodology to the Development of Chemoselective Ligations for Bioorganic Applications

Cyrille Sabot
Advances in Chemical Sciences and Technologies (ACST, 2019), Sep 2019, Warangal, India
Conference papers hal-02372314v1

Fast-Responsive Nitroso-Based Turn-On Probe for Hydrogen Sulfide

Kévin Renault , Cyrille Sabot , Pierre-Yves Renard
European Journal of Organic Chemistry, 2015, 2015 (36), pp.7992-7996. ⟨10.1002/ejoc.201501140⟩
Journal articles istex hal-02046170v1
Image document

Fluorophore-assisted click chemistry through copper(I) complexation

Victor Flon , Magalie Bénard , Damien Schapman , Ludovic Galas , Pierre-Yves Renard , et al.
Biomolecules, 2020, 10 (4), pp.619. ⟨10.3390/biom10040619⟩
Journal articles hal-03034414v1