Crystal structures ofLymphocytic choriomeningitis virusendonuclease domain complexed with diketo-acid ligands
Magali Saez-Ayala
,
Elsie Yekwa
,
Mauro Carcelli
,
Bruno Canard
,
Karine Alvarez
,
et al.
Journal articles
hal-03078366v1
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Synthesis and Anti-BVDV Activity of Acridones As New Potential Antiviral Agents 1
Oriana Tabarrini
,
Giuseppe Manfroni
,
Arnaldo Fravolini
,
Violetta Cecchetti
,
Stefano Sabatini
,
et al.
Journal articles
istex
hal-02459231v1
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Structural Analysis of the Activation of Ribavirin Analogs by NDP Kinase: Comparison with Other Ribavirin Targets
Sarah Gallois-Montbrun
,
Yuxing Chen
,
Hélène Dutartre
,
Magali Sophys
,
Solange Moréra
,
et al.
Journal articles
hal-02459258v1
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The Imidazopyrrolopyridine Analogue AG110 Is a Novel, Highly Selective Inhibitor of Pestiviruses That Targets the Viral RNA-Dependent RNA Polymerase at a Hot Spot for Inhibition of Viral Replication
Jan Paeshuyse
,
Jean-Michel Chezal
,
Matheus Froeyen
,
Pieter Leyssen
,
Hélène Dutartre
,
et al.
Journal articles
hal-02459217v1
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Gln151 of HIV-1 reverse transcriptase acts as a steric gate towards clinically relevant acyclic phosphonate nucleotide analogues.
Antoine Frangeul
,
Cécile Bussetta
,
Jérôme Deval
,
Karine Barral
,
Karine Alvarez
,
et al.
Antiviral Therapy , 2019, 13 (1), pp.115-24
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hal-02061712v1
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In Vitro Suppression of K65R Reverse Transcriptase-Mediated Tenofovir- and Adefovir-5'-Diphosphate Resistance Conferred by the Boranophosphonate Derivatives
A. Frangeul
,
Karine Barral
,
K. Alvarez
,
B. Canard
Journal articles
hal-02061675v1
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Substrate selectivity of Dengue and Zika virus NS5 polymerase towards 2′-modified nucleotide analogues
Supanee Potisopon
,
Francois Ferron
,
Véronique Fattorini
,
Barbara Selisko
,
Bruno Canard
Journal articles
hal-01802946v1
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Alkylated flavanones from the bark of Cryptocarya chartacea as dengue virus NS5 polymerase inhibitors.
Pierre-Marie Allard
,
Elise Tran Huu Dau
,
Cécilia Eydoux
,
Jean-Claude Guillemot
,
Vincent Dumontet
,
et al.
Journal articles
hal-00684627v1
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The viral capping enzyme nsP1: a novel target for the inhibition of chikungunya virus infection
L. Delang
,
C. Li
,
A. Tas
,
G. Querat
,
I. C. Albulescu
,
et al.
Journal articles
hal-01439113v1
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SPINE bioinformatics and data-management aspects of high-throughput structural biology.
S. Albeck
,
Pedro Maria Alzari
,
C. Andreini
,
L. Banci
,
I. M. Berry
,
et al.
Journal articles
hal-00187834v1
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Biodiversity as a source of potent and selective inhibitors of Chikungunya virus replication
Pieter Leyssen
,
Jacqueline Smadja
,
Philippe Rasoanaivo
,
Ameenah Gurib-Fakim
,
Mohamad Fawzi-Mahomoodally
,
et al.
Gurib-Fakim, A.
Novel Plant Bioresources, Applications in Food, Medicine and Cosmetics, , John Wiley & Sons, Ltd, Chichester UK., pp.151-160, 2014, 978-1-118-46061-0.
⟨10.1002/9781118460566.ch11⟩
Book sections
hal-01163238v1
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Metal chelators for the inhibition of the lymphocytic choriomeningitis virus endonuclease domain
Magali Saez-Ayala
,
Elsie Laban Yekwa
,
Clémence Mondielli
,
Loic Roux
,
Sergio Hernández
,
et al.
Journal articles
hal-03076409v1
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Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication
Karine Barral
,
Clément Weck
,
Nadine Payrot
,
Loic Roux
,
Céline Durafour
,
et al.
Journal articles
hal-02061721v1
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Expression, purification and crystallization of the SARS-CoV macro domain
Hélène Malet
,
Karen Dalle
,
Nicolas Bremond
,
Fabienne Tocque
,
Stéphanie Blangy
,
et al.
Acta Crystallographica Section F: Structural Biology and Crystallization Communications , 2006, 62 (4), pp.405-408.
⟨10.1107/S1744309106009274⟩
Journal articles
hal-02066254v1
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Coronavirus Nsp10, a critical co-factor for activation of multiple replicative enzymes
Mickaël Bouvet
,
Adrien Lugari
,
Clara C. Posthuma
,
Jessika C. Zevenhoven
,
Stéphanie Bernard
,
et al.
Journal articles
hal-01910944v1
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Structural and Functional Basis of the Fidelity of Nucleotide Selection by Flavivirus RNA-Dependent RNA Polymerases
Barbara Selisko
,
Nicolas Papageorgiou
,
Francois Ferron
,
Bruno Canard
Journal articles
hal-02094550v1
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Observation of arenavirus nucleoprotein heptamer assembly
Nicolas Papageorgiou
,
Afroditi Vaitsopoulou
,
Awa Diop
,
Thi Hong van Nguyen
,
Bruno Canard
,
et al.
Journal articles
hal-03143071v1
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Flacourtosides A-F, Phenolic Glycosides Isolated from Flacourtia ramontchi.
Mélanie Bourjot
,
Pieter Leyssen
,
Cécilia Eydoux
,
Jean-Claude Guillemot
,
Bruno Canard
,
et al.
Journal articles
hal-00694429v1
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Filovirus proteins for antiviral drug discovery: Structure/function bases of the replication cycle
Baptiste Martin
,
Bruno Canard
,
Etienne Decroly
Journal articles
hal-01802809v1
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Development of specific dengue virus 2'-O- and N7-methyltransferase assays for antiviral drug screening.
Karine Barral
,
Corinne Sallamand
,
Christiane Petzold
,
Bruno Coutard
,
Axelle Collet
,
et al.
Journal articles
hal-00874640v1
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Primer-Dependent and Primer-Independent Initiation of Double Stranded RNA Synthesis by Purified Arabidopsis RNA-Dependent RNA Polymerases RDR2 and RDR6
Anthony Devert
,
Nicolas Fabre
,
Maïna Floris
,
Bruno Canard
,
Christophe Robaglia
,
et al.
Journal articles
hal-01217572v1
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Rapid incorporation of Favipiravir by the fast and permissive viral RNA polymerase complex results in SARS-CoV-2 lethal mutagenesis
Ashleigh Shannon
,
Barbara Selisko
,
Nhung-Thi-Tuyet Le
,
Johanna Huchting
,
Franck Touret
,
et al.
Journal articles
inserm-03052188v1
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Snapshots of ADp-ribose bound to Getah virus macro domain reveal an intriguing choreography
Ana Sofia Ferreira-Ramos
,
Gerlind Sulzenbacher
,
Bruno Canard
,
Bruno Coutard
Journal articles
hal-03160433v1
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Drugs against SARS‐CoV ‐2: What do we know about their mode of action?
Coralie Valle
,
Baptiste Martin
,
Franck Touret
,
Ashleigh Shannon
,
Bruno Canard
,
et al.
Journal articles
hal-03030758v1
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The methyltransferase domain of the Respiratory Syncytial Virus L protein catalyzes cap N7 and 2’-O-methylation
Priscila Sutto-Ortiz
,
Sergey Tcherniuk
,
Nina Ysebaert
,
Pravien Abeywickrema
,
Mathieu Noël
,
et al.
Journal articles
hal-03352803v1
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Chemical constituents of Anacolosa pervilleana and their antiviral activities.
Mélanie Bourjot
,
Pieter Leyssen
,
Cécilia Eydoux
,
Jean-Claude Guillemot
,
Bruno Canard
,
et al.
Journal articles
istex
hal-00722062v1
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Preparation of purine and pyrimidine acyclic nucleotide analogs as antiviral agents
Karine Barral
,
Bruno Canard
,
Karine Alvarez
,
Jean-Louis Romette
,
Johan Neyts
,
et al.
France, Patent n° : WO 2007-IB4233. 2007
Patents
hal-02063281v1
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The Curious Case of the Nidovirus Exoribonuclease: Its Role in RNA Synthesis and Replication Fidelity
Natacha S Ogando
,
Francois Ferron
,
Etienne Decroly
,
Bruno Canard
,
Clara C Posthuma
,
et al.
Journal articles
hal-02353805v1
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The Crystal Structures of Chikungunya and Venezuelan Equine Encephalitis Virus nsP3 Macro Domains Define a Conserved Adenosine Binding Pocket
H. Malet
,
B. Coutard
,
S. Jamal
,
H. Dutartre
,
N. Papageorgiou
,
et al.
Journal articles
hal-02459209v1
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Acyclic phosphonate nucleotides and human adenylate kinases: impact of a borano group on alpha-P position.
D. Topalis
,
K. Alvarez
,
K. Barral
,
Hélène Munier-Lehmann
,
B. Schneider
,
et al.
Journal articles
pasteur-00316017v1
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