Structure-Based Design and Biological Characterization of Selective Histone Deacetylase 8 (HDAC8) Inhibitors with Anti-Neuroblastoma Activity
Tino Heimburg
(1)
,
Fiona Kolbinger
,
Patrik Zeyen
,
Ehab Ghazy
,
Daniel Herp
,
Karin Schmidtkunz
(2)
,
Jelena Melesina
(1)
,
Tajith Baba Shaik
,
Frank Erdmann
,
Matthias Schmidt
,
Christophe Romier
(3)
,
Dina Robaa
(1)
,
Olaf Witt
(4)
,
Ina Oehme
,
Manfred Jung
,
Wolfgang Sippl
(5)
1
MLU -
Martin-Luther-Universität Halle Wittenberg
2 Albert-Ludwigs-Universität Freiburg
3 IGBMC - Institut de Génétique et de Biologie Moléculaire et Cellulaire
4 Department of Pediatric Oncology, Hematology and Immunology, Heidelberg University Hospital, Heidelberg, Germany
5 Institute of Pharmaceutical Chemistry
2 Albert-Ludwigs-Universität Freiburg
3 IGBMC - Institut de Génétique et de Biologie Moléculaire et Cellulaire
4 Department of Pediatric Oncology, Hematology and Immunology, Heidelberg University Hospital, Heidelberg, Germany
5 Institute of Pharmaceutical Chemistry
Tino Heimburg
- Function : Author
- PersonId : 795732
- ORCID : 0000-0002-8400-7191
Fiona Kolbinger
- Function : Author
Patrik Zeyen
- Function : Author
Ehab Ghazy
- Function : Author
Daniel Herp
- Function : Author
Tajith Baba Shaik
- Function : Author
Frank Erdmann
- Function : Author
- PersonId : 798761
- ORCID : 0000-0001-5261-0984
Matthias Schmidt
- Function : Author
Christophe Romier
- Function : Author
- PersonId : 750418
- IdHAL : christophe-romier
- ORCID : 0000-0002-3680-935X
- IdRef : 161229859
Ina Oehme
- Function : Author
Manfred Jung
- Function : Author
Wolfgang Sippl
- Function : Author
- PersonId : 761816
- ORCID : 0000-0002-5985-9261
- IdRef : 067715265